| VCB | 维库溴铵 | Vecuronium bromide | 50700-72-6 |
| MAB | 马波沙星 | MARBOFLOXACIN | 115550-35-1 |
| MAB01 | 6,8-二氟-1-(甲酰基甲基氨基)-7-(4-甲基-1-哌嗪基)-4-氧代-1,4-二氢喹啉-3-甲酸乙酯 | 6,8-Difluoro-1-(formylmethylamino)-7-(4-methylpiperazin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid ethyl ester | 158585-86-5 |
| MAB02 | 6,7,8-三氟-1-(甲酰基甲基氨基)-4-氧代-1,4-二氢喹啉-3-甲酸乙酯 | 6,7,8-Trifluoro-1-(formylmethylamino)-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid ethyl ester | 100276-65-1 |
| IT | 依鲁替尼 | Ibrutinib | 936563-96-1 |
| IT01 | 依鲁替尼N-1 | 3-(4-Phenoxy-phenyl)-1-piperidin-3-yl-1H-pyrazolo[3,4-d]pyriMidin-4-ylaMine | 1022150-12-4 |
| IT02 | (R)-3-[4-氨基-3-(4-苯氧基苯基)-1H-吡唑并[3,4-D]嘧啶-1-基]哌啶-1-羧酸叔丁酯 | 3-[4-Amino-3-(4-phenoxy-phenyl)-pyrazolo[3,4-d]pyrimidin-1-yl]-piperidine-1-carboxylic acid tert-butyl ester | 1022150-11-3 |
| IT03 | 3-(4-苯氧基苯基)-1H- 吡唑并[3,4-D]嘧啶-4-胺 | 5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyriMidin-4-ylaMine | 330786-24-8 |
| IT04 | (S)-1-叔丁氧羰基-3-羟基哌啶 | (S)-1-Boc-3-hydroxypiperidine | 143900-44-1 |
| IT05 | 3-(4-苯氧基苯基)-1-(3R)-3-哌啶基-1H-吡唑并[3,4-D]嘧啶-4-胺盐酸盐(1:2) | (R)-3-(4-phenoxyphenyl)-1-(piperidin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine dihydrochloride | 1701403-10-2 |
| IT06 | 2-[(羟基)(4-苯氧基苯基)亚甲基]丙二腈 | 2-[Hydroxy-(4-phenoxy-phenyl)-Methylene]-Malononitrile | 330792-68-2 |
| OPB | 奥拉帕尼 | Olaparib | 763113-22-0 |
| NT | 奈妥吡坦 | Netupitant | 290297-26-6 |
| NT01 | 2-(3,5-二(三氟甲基)苯基)-2-甲基丙酸 | 2-[3,5-bis(trifluoromethyl)phenyl]-2-methylpropanoic acid | 289686-70-0 |
| NT02 | 奈妥吡坦中间体2 | [6-(4-methyl-piperazin-1-yl)-4-o-tolylpyridin-3-yl]-carbamic | 342417-02-1 |
| NT03 | 奈妥吡坦N-1 | methyl-[6-(4-methyl-piperazin-1-yl)-4-o-tolyl-pyridin-3-yl]-amine | 290297-25-5 |
| NT04 | 6-(4-甲基哌嗪-1-基)-4-(2-甲基苯基)烟酰胺 | 4-(2-methylphenyl)-6-(4-methylpiperazin-1-yl)pyridine-3-carboxamide | 342417-01-0 |
| NT05 | N-叔丁基-6-氯-4-邻甲苯基烟酰胺 | N-tert-butyl-6-chloro-4-(o-tolyl)nicotinamide | 342417-04-3 |
| AZD | AZD-9291,甲磺酸-迈瑞替尼 | AZD-9291 (Mesylate) | 1421373-66-1 |
| AZD001 | 4-氟-2-甲氧基-5-硝基苯胺 | 4-Fluoro-2-methoxy-5-nitroaniline | 1075705-01-9 |
| AZD002 | N1-[2-(二甲基氨基)乙基]-5-甲氧基-N1-甲基-N4-[4-(1-甲基-1H-吲哚-3-基)-2-嘧啶基]-1,2,4-苯三胺 | N1-(2-(dimethylamino)ethyl)-5-methoxy-N1-methyl-N4-(4-(1-methyl-1H-indol-3-yl)pyrimidin-2-yl)benzene-1,2,4-triamine | 1421372-66-8 |
| AZD003 | 3-(2-氯-4-嘧啶基)-1-甲基-1H-吲哚 | 3-(2-chloropyrimidin-4-yl)-1-methylindole | 1032452-86-0 |
| AZD004 | N-(4-氟-2-甲氧基-5-硝基苯基)-4-(1-甲基-1H-吲哚-3-基)-2-嘧啶胺 | N-(4-Fluoro-2-methoxy-5-nitrophenyl)-4-(1-methyl-1H-indol-3-yl)-2-pyrimidinamine | 1421372-94-2 |
| AZD005 | N-(2-二甲基氨基-乙基)-2-甲氧基-n-甲基-n-[4-(1-甲基-1H-吲哚-3-基)-嘧啶-2-基]-5-硝基-苯-1,4-二胺 | N1-(2-(dimethylamino)ethyl)-5-methoxy-N1-methyl-N4-(4-(1-methyl-1H-indol-3-yl)pyrimidin-2-yl)-2-nitrobenzene-1,4-diamine | 1421372-67-9 |
| FVST | 氟维司群 | Fulvestrant | 129453-61-8 |
| FVST02 | (7A,17B)- 7-(9-溴壬基)雌甾-1,3,5(10)-三烯-3,17-二醇 | (7a,17b)-7-(9-Bromononyl)estra-1,3,5(10)-triene-3,17-diol | 875573-67-4 |
| FVST03 | (7A,17B)-7-(9-溴壬基)雌甾-1,3,5(10)-三烯-3,17-二醇 17-醋酸酯 | (7a,17b)-7-(9-Bromononyl)-estra-1,3,5(10)-triene-3,17-diol 17-acetate | 875573-66-3 |
| FD | 福沙匹坦二甲葡胺 | Fosaprepitant dimeglumine | 265121-04-8 |
| CB | 乙酸阿比特龙酯 | Abiraterone acetate | 154229-18-2 |
| CB01 | 阿比特龙 | Abiraterone | 154229-19-3 |
| CB02 | 17-碘雄甾-5,16-二烯-3β-醇 | 17-Iodoandrosta-5,16-dien-3beta-ol | 32138-69-5 |
| SLN | 塞利尼索 | Selinexor | 1393477-72-9 |
| SLN01 | 3-(3,5-双(三氟甲基)苯基)-1H-1,2,4-三唑 | 3-(3,5-bis(trifluoroMethyl)phenyl)-1H-1,2,4-triazole | 1333154-10-1 |
| SLN02 | (Z)-3-(3-(3,5-双(三氟甲基)苯基)-1H-1,2,4-三唑-1-基)丙烯酸 | (Z)-3-(3-(3,5-bis(trifluoromethyl)phenyl)-1H- 1,2,4-triazol-1-yl)acrylic acid | 1388842-44-1 |
| SLN03 | (Z)-3-(3-(3,5-双(三氟甲基)苯基)-1H-1,2,4-三唑-1-基)丙烯酸异丙酯 | (Z)-isopropyl 3-(3-(3,5-bis(trifluoromethyl)phenyl)-1H-1,2,4-triazol-1-yl)acrylate | 1333152-22-9 |
| SLN04 | (Z)异丙基丙烯酸异丙酯 | (Z)-ISOPROPYL 3-IODOACRYLATE | 1333154-26-9 |
| SLN05 | 丙炔酸异丙酯 | 2-Propynoic acid | 96088-62-9 |
| PRBL | 普瑞巴林 | Pregabalin | 148553-50-8 |
| LD | 雷迪帕韦 | Ledipasvir,GS5885 | 1256388-51-8 |
| LD01 | 雷迪帕韦丙酮盐 | Ledipasvir (acetone) | 1441674-54-9 |
| LD03 | (S)-5-(叔丁氧羰基)-5-氮杂螺[2.4]庚烷-6-羧酸 | (S)-5-(tert-Butoxycarbonyl)-5-azaspiro[2.4]heptane-6-carboxylic acid | 1129634-44-1 |
| LD04 | (S)-5-(叔丁氧羰基)-5-氮杂螺[2.4]庚烷-6-羧酸钾 | (6S)-5-Azaspiro[2.4]heptane-5,6-dicarboxylic acid 5-(1,1-diMethylethyl) ester potassiuM salt | 1441673-92-2 |
| LD05 | 1-(7-溴-9,9-二氟-9H-芴-2-基)-2-氯乙酮 | 1-(7-broMo-9,9-difluoro-9H-fluoren-2-yl)-2-chloro-Ethanone | 1378387-81-5 |
| LD06 | (1R,3S,4S)-3-(6-溴-1H-苯并咪唑-2-基)-2-氮杂双环[2.2.1]庚烷-2-羧酸叔丁酯
| 2-Azabicyclo[2.2.1]heptane-2-carboxylic acid | 1256387-74-2 |
| LD07 | (1R,3S,4S)-2-(叔丁氧羰基)- 3-(6-(硼酸频哪醇酯)-1H-苯并[D]咪唑-2-基)-2-氮杂双环[2.2.1]庚烷 | (1R,3S,4S)-tert-butyl 3-(6-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-benzo[d]iMidazol-2-yl)-2-azabicyclo[2.2.1]heptane-2-carboxylate | 1256387-87-7 |
| LD08 | (S)-5 -叔丁氧羰基-6-(5 - (7 - 溴-9,9-二氟-9H-芴-2-基)-1H-咪唑-2-基)-5-氮杂螺[2.4]庚烷 | (S)-tert-butyl 6-(5-(7-broMo-9,9-difluoro-9H-fluoren-2-yl)-1H-iMidazol-2-yl)-5-azaspiro[2.4]heptane-5-carboxylate | 1441670-89-8 |
| VPSR | 维帕他韦 | Velpatasvir | 1377049-84-7 |
| SF | 索非布韦 | sofosbuvir | 1190307-88-0 |
| SF01 | 索菲布韦中间体 | ((2R,3R,4R)-3-(benzoyloxy)-4-fluoro-4-methyl-5-oxotetrahydrofuran-2-yl)methyl benzoate | 874638-80-9 |
| TAK-438 | 氟呐普拉赞 | TAK-438,Vonoprazan FuMarate | 881681-01-2;1260141-27-2 |
| TAK-43801 | 吡啶-3-磺酰氯 | 3-Pyridinesulfonyl chloride | 16133-25-8; 813222-82-1 |
| TAK-43802 | 5-(2-氟苯基)-1H-吡咯-3-甲醛 | 5-(2-fluorophenyl)-1H-pyrrole-3-carbaldehyde | 881674-56-2 |
| BA | 布瓦西坦 | Brivaracetam | 357336-20-0 |
| BA01 | (R)-4-丙基-二氢呋喃-2-酮 | (R)-4-Propyldihydrofuran-2(3H)-one | 63095-51-2 |
| OA | 奥贝胆酸 | 6-Ethylchenodeoxycholic acid | 459789-99-2 |
| OA01 | 3Α-羟基-7-氧代-5Β-胆烷酸 | 3-alpha-hydroxy-7-oxo-5-beta-cholan-24-oic acid | 4651-67-6 |
| OA04 | 3A-羟基-6-乙叉基-7-氧代-24-胆烷酸 | Obeticholic Acid-G | 1516887-33-4 |
| AB | 阿维巴坦钠 | avibactam sodium | 1192491-61-4 |
| AB01 | 阿维巴坦四丁基铵盐 | N,N,N-tributyl-1-Butanaminium (1R,2S,5R)-2-(aminocarbonyl)-7-oxo-1,6-diazabicyclo[3.2.1]oct-6-yl sulfate | 1192651-80-1 |
| AB02 | 阿维巴坦 | avibactam | 1192500-31-4 |
| AB03 | (2S,5R)-苯氧胺基哌啶-2-甲酰胺 | (2S,5R)-5-[(benzyloxy)amino]piperidine-2-carboxamide | 1416134-49-0 |
| AB04 | 阿维巴坦钠中间体1;(2S,5R)-苯氧胺基哌啶-2-甲酸乙酯草酸盐 | (2S, 5R) -benzyloxyaminopiperidine-2-carboxylic acid ethyl oxalate | 1416134-48-9 |
| AB05 | (2S,5R)-6-(苄氧)-7-氧-1,6-二氮杂二环[3.2.1]辛烷-2-甲酰胺 | (2S,5R)-6-(benzyloxy)-7-oxo-1,6-diazabicyclo[3.2.1]octane-2-carboxamide | 1192651-49-2 |
| AG | 苯甲酸阿格列汀 | 2-[6-[3(R)-Aminopiperidin-1-yl]-3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-ylmethyl]benzonitrile benzoate | 850649-62-6 |
| AG01 | (R)-3-氨基哌啶双盐酸盐 | (R)-3-AMINOPIPERIDINE DIHYDROCHLORIDE | 334618-23-4 |
| TC | 枸橼酸托法替布 | Tofacitinib citrate | 540737-29-9 |
| TC01 | 托法替布 | Tofacitinib | 477600-75-2 |
| TC02 | (3R,4R)-1-苄基-N,4-二甲基哌啶-3-胺二盐酸盐 | (3R,4R)-N,4-Dimethyl-1-(phenylmethyl)-3-piperidinamine hydrochloride | 1062580-52-2 |
| TC03 | 2,4-二氯-1H-吡咯并[2,3-d]嘧啶 | 2,4-Dichloro-1H-pyrrolo[2,3-d]pyrimidine | 90213-66-4 |
| RMTN | 雷美替胺 | Ramelteon | 196597-26-9 |
| RMTN01 | (S)-2-(1,6,7,8-四氢-2H-茚并(5,4-b)呋喃-8-基)乙胺 | (S)-2-(1,6,7,8-Tetrahydro-2H-indeno[5,4-b]furan-8-yl)ethylamine | 196597-81-6 |
| RMTN02 | 1,2,6,7-四氢-8H-茚并[5,4-b]呋喃-8-酮 | 1,2,6,7-Tetrahydro-8H-indeno[5,4-b]furan-8-one | 196597-78-1 |
| APST | S)-2-[1-(3-乙氧基-4-甲氧基苯基)-2-甲磺酰基乙基]-4-乙酰基氨基异吲哚啉-1,3-二酮 | Apremilast | 608141-41-9 |
| APST01 | 3-乙酰氨基邻苯二甲酸酐 | 1,3-Dioxo-2-isoindolineaceticacid | 6296-53-3 |
| APST02 | (S)-1-(3-乙氧基-4-甲氧基苯基)-2-(甲基磺酰基)乙胺 N-乙酰基-L-亮氨酸盐 | (S)-1-(3-Ethoxy-4-Methoxyphenyl)-2-(Methylsulfonyl)ethylaMine N-acetyl-L-leucine salt | 608141-43-1 |
| MK310201 | 2-(甲基磺酰基)-2,6-二氢吡咯并[3,4-c]吡唑-5(4H)-羧酸叔丁酯 | tert-butyl 2-(Methylsulfonyl)-4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate | 1226781-82-3 |
| MK310202 | 2-(甲基磺酰基)-2,4,5,6-四氢吡咯并[3,4-c]吡唑 苯磺酸盐 | 2-(Methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole | 1280210-80-1 |
| MK310203 | ((2R,3S)-2-(2,5-二氟苯基)-3,4-二氢-2H-吡喃-3-基)氨基甲酸叔丁酯 | tert-butyl [(2R,3S)-2-(2,5-difluorophenyl)-3,4-dihydro-2H-pyran-3-yl]carbaMate | 1172623-98-1 |
| MK310204 | N-[(2R,3S)-2-(2,5-二氟苯基)四氢-5-氧-2H-吡喃-3-基]-氨基甲酸 1,1-二甲基乙基酯 | N-[(2R,3S)-2-(2,5-difluorophenyl)tetrahydro-5-oxo-2H-pyran-3-yl]-CarbaMic acid 1,1-diMethylethyl ester | 951127-25-6 |
| SRFN | 索拉非尼 | Sorafenib | 284461-73-0 |
| SRFN01 | 4-氯-3-(三氟甲基)苯异氰酸酯 | 4-Chloro-3-(trifluoromethyl)phenyl isocyanate | 327-78-6 |
| SRFN02 | N-甲基-4-氯-2-吡啶甲酰胺 | N-Methyl-4-chloropyridine-2-carboxamide | 220000-87-3 |
| SRFN03 | 4-(4-氨基苯氧基)-N-甲基-2-吡啶甲酰胺 | 4-(4-Aminophenoxy)-N-methylpicolinamide | 284462-37-9 |
| AP | AP26113 | 5-chloro-2-N-[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl]-4-N-(2-dimethylphosphorylphenyl)pyrimidine-2,4-diamine | 1197958-12-5 |
| GS | 替诺福韦艾拉酚胺半富马酸盐 | Tenofovir Alafenamide Fumarate | 1392275-56-7 |
| IDB | 靛玉红 | Indirubin | 479-41-4 |
| IDB01 | 3-吲哚乙酸酚酯 | 3-ACETOXYINDOLE | 608-08-2 |
| RBAP | (R)-3-叔丁氧羰基氨基哌啶 | (R)-3-(Boc-Amino)piperidine | 309956-78-3 |
| BTXB | 贝曲西班马来酸盐 | Betrixaban maleate | 936539-80-9 |
| BTXB01 | 贝曲西班 | Betrixaban | 330942-05-7 |
| BTXB02 | N-(5-氯-2-吡啶)-5-甲氧基-2-氨基苯甲酰胺 | 2-AMino-N-(5-chloropyridin-2-yl)-5-MethoxybenzaMide | 280773-17-3 |
| DLXC | 德拉沙星 | Delafloxacin | 189279-58-1 |
| DLXCM | 德拉沙星葡甲胺盐 | Delafloxacin (MegluMine) | 352458-37-8 |
| DLXC01 | 2,6-二氨基-3,5-二氟嘧啶 | 3,5-Difluoropyridine-2,6-diamine | 247069-27-8 |
| DLXC02 | 2,4,5-三氟苯甲酰乙酸乙酯 | 2,4,5-Triflurobenzoflacetate | 98349-24-7 |
| DLXC03 | 3-羟基氮杂环丁二烯盐酸盐 | 3-Hydroxyazetidine hydrochloride | 18621-18-6 |
| DLXC04 | 2,3,5,6-四氟吡啶 | 2,3,5,6-Tetrafluoropyridine | 2875-18-5 |
| LCZ696 | LCZ696 | LCZ 696 | 936623-90-4 |
| LCZ696-01 | AHU-377 钙盐 | AHU-377 (heMicalciuM salt) | 1369773-39-6 |
| LCZ696-02 | AHU-377 | 4-(((2R,4R)-1-([1,1'-biphenyl]-4-yl)-5-ethoxy-4-Methyl-5-oxopentan-2-yl)aMino)-4-oxobutanoic acid | 149709-62-6 |
| LCZ696-03 | N-[(1R)-2-[1,1'-联苯]-4-基-1-(羟基甲基)乙基]氨基甲酸叔丁酯 | N-[(1R)-2-[1,1'-Biphenyl]-4-yl-1-(hydroxymethyl)ethyl]carbamic acid 1,1-dimethylethyl ester | 1426129-50-1 |
| LCZ696-04 | (2R,4S)-5-(联苯-4-基)-4-[(叔丁氧基羰基)氨基]-2-甲基戊酸 | (2R,4S)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)aMino)-2-Methylpentanoic acid | 1012341-50-2 |
| IZ | 艾沙康唑 | Isavuconazole | 241479-67-4 |
| IZ01 | 艾沙康唑硫酸盐 | Isavuconazonium sulfate | 946075-13-4 |
| IZ02 | 4-溴乙酰基苯腈 | 4-Cyanophenacyl bromide | 20099-89-2 |
| IZ03 | (2R, 3R)-3-(2, 5-二氟苯基)-3-羟基-2-甲基-4-[1H-(1, 2, 4)-三氮唑-1-基]硫代丁酰胺 | (2R,3R)-3-(2,5-Difluorophenyl)-3-hydroxy-2-Methyl-4-(1H-1,2,4-triazol-1-yl)thiobutyraMide | 368421-58-3 |
| IZ04 | (2S,3R)- 3-(2,5-二氟)-3-羟基-2-甲基-4-(1H-1,2,4-三唑-1-基)丁腈 | (αS,βR)-β-(2,5-Difluorophenyl)-β-hydroxy-α-Methyl-1H-1,2,4-triazole-1-butanenitrile | 241479-74-3 |
| IZ05 | 4-氰基-1-(2,6-二氟苄基)-1H-1,2,3-三氮唑 | 1-[[(2R,3S)-2-(2,5-Difluorophenyl)-3-methyloxiranyl]methyl]-1H-1,2,4-triazole | 241479-73-2 |
| IZ06 | N-甲基-N-(3-[((N-叔丁氧羰基-N-甲基氨基)乙酰氧基)甲基]吡啶-2-基)氨基甲酸(1-氯乙基)酯 | Glycine, N-[(1,1-diMethylethoxy)carbonyl]-N-Methyl-, [2-[[(1-chloroethoxy)carbonyl]MethylaMino]-3-pyridinyl]Methyl ester | 338990-31-1 |
| IZ07 | 艾沙康唑侧链中间体2 | 2-(methylamino)pyridin-3-yl)methyl 2-((tert-butoxycarbonyl)(methyl)amino)acetate | 1180002-01-0 |
| IZ08 | 2-甲胺基-3-吡啶甲醇 | 2-(Methylamino)pyridine-3-methanol | 32399-12-5 |
| EFZ | 艾氟康唑 | Efinaonazole | 164650-44-6 |
| EFZ01 | 1-(((2R,3S),2-(2,4-二氟苯基)-3-甲基环氧乙烷-2-基)甲基)-1H-1,2,4-三唑 | 1-(((2R,3S)-2-(2,4-Difluorophenyl)-3-methyloxiran-2-yl) methyl)-1H-1,2,4-triazole | 127000-90-2 |